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Summary on some antiviral researches

1. Niclosamide:    Mode of Action:  Neutralization of endosomal pH *Also affects maturation of Dengue virus (DENV) particles rendering them non-infectious (1).   *It is an antiparasitic   drug approved drug for human use.  2.  1-methylpropyl-2-imidazolyl disulfide (PX-12):      Mode of Action:    Reversible inhibition of the thioredoxin system (Trx1 system) causing a slow irreversible thioalkylation of Trx1  (2) .  *Anti-HIV-1 effect. In hibited the enzymatic activity of Trx1 and the Trx1-dependent disulfide reduction of gp120.   *Developed as an antitumor agent. 3.    Nitazoxanide (NTZ):    Mode of Action:  Inhibits host ERp57 activity, causing newly synthesized F-protein misfolding, F-aggregate formation and halting F-trafficking to the host plasma membrane as reported in a prototype    paramyxovirus Sendai (SeV) (3).  ...